Discovery, Modeling, and Human Pharmacokinetics of N-(2-Acetyl-4,6-dimethylphenyl)-3-(3,4-dimethylisoxazol-5-ylsulfamoyl) -thiophene-2-carboxamide (TBC3711), a Second Generation, ETA Selective, and Orally Bioavailable Endothelin Antagonist

Chengde Wu, E. Radford Decker, Natalie Blok, Huong Bui, Tony J. You, Junmei Wang, Andree R. Bourgoyne, Vippra Knowles, Kurt L. Berens, George W. Holland, Tommy A. Brock, Richard A F Dixon

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