Discovery of 3α,7α,11β-Trihydroxy-6α-ethyl-5β-cholan-24-oic Acid (TC-100), a Novel Bile Acid as Potent and Highly Selective FXR Agonist for Enterohepatic Disorders

Roberto Pellicciari, Daniela Passeri, Francesca De Franco, Serena Mostarda, Paolo Filipponi, Carolina Colliva, Raffaella Maria Gadaleta, Placido Franco, Andrea Carotti, Antonio Macchiarulo, Aldo Roda, Antonio Moschetta, Antimo Gioiello

Research output: Contribution to journalArticlepeer-review

47 Scopus citations

Fingerprint

Dive into the research topics of 'Discovery of 3α,7α,11β-Trihydroxy-6α-ethyl-5β-cholan-24-oic Acid (TC-100), a Novel Bile Acid as Potent and Highly Selective FXR Agonist for Enterohepatic Disorders'. Together they form a unique fingerprint.

Chemical Compounds

Medicine & Life Sciences