Fused tetrazoles as azide surrogates in click reaction: Efficient synthesis of N-heterocycle-substituted 1,2,3-triazoles

Buddhadeb Chattopadhyay; Claudia I.Rivera Vera; Stepan Chuprakov; Vladimir Gevorgyan

doi:10.1021/ol100745d

Fused tetrazoles as azide surrogates in click reaction: Efficient synthesis of N-heterocycle-substituted 1,2,3-triazoles

Buddhadeb Chattopadhyay, Claudia I.Rivera Vera, Stepan Chuprakov, Vladimir Gevorgyan

Research output: Contribution to journal › Article › peer-review

100 Scopus citations

Abstract

Figure presented It has been shown that various pyrido-, quinolino-, pyrazino-, and quinoxalinotetrazoles can be used efficiently as azide components in Cu-catalyzed click reaction with alkynes. This method allows for efficient synthesis of a wide variety of N-heterocyclic derivatives of 1,2,3-triazoles.

Original language	English (US)
Pages (from-to)	2166-2169
Number of pages	4
Journal	Organic Letters
Volume	12
Issue number	9
DOIs	https://doi.org/10.1021/ol100745d
State	Published - May 7 2010
Externally published	Yes

ASJC Scopus subject areas

Biochemistry
Physical and Theoretical Chemistry
Organic Chemistry

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10.1021/ol100745d

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abstract = "Figure presented It has been shown that various pyrido-, quinolino-, pyrazino-, and quinoxalinotetrazoles can be used efficiently as azide components in Cu-catalyzed click reaction with alkynes. This method allows for efficient synthesis of a wide variety of N-heterocyclic derivatives of 1,2,3-triazoles.",

author = "Buddhadeb Chattopadhyay and Vera, {Claudia I.Rivera} and Stepan Chuprakov and Vladimir Gevorgyan",

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T1 - Fused tetrazoles as azide surrogates in click reaction

T2 - Efficient synthesis of N-heterocycle-substituted 1,2,3-triazoles

AU - Chattopadhyay, Buddhadeb

AU - Vera, Claudia I.Rivera

AU - Chuprakov, Stepan

AU - Gevorgyan, Vladimir

PY - 2010/5/7

Y1 - 2010/5/7

N2 - Figure presented It has been shown that various pyrido-, quinolino-, pyrazino-, and quinoxalinotetrazoles can be used efficiently as azide components in Cu-catalyzed click reaction with alkynes. This method allows for efficient synthesis of a wide variety of N-heterocyclic derivatives of 1,2,3-triazoles.

AB - Figure presented It has been shown that various pyrido-, quinolino-, pyrazino-, and quinoxalinotetrazoles can be used efficiently as azide components in Cu-catalyzed click reaction with alkynes. This method allows for efficient synthesis of a wide variety of N-heterocyclic derivatives of 1,2,3-triazoles.

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M3 - Article

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JO - Organic Letters

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Fused tetrazoles as azide surrogates in click reaction: Efficient synthesis of N-heterocycle-substituted 1,2,3-triazoles

Abstract

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