Fused tetrazoles as azide surrogates in click reaction: Efficient synthesis of N-heterocycle-substituted 1,2,3-triazoles

Buddhadeb Chattopadhyay, Claudia I.Rivera Vera, Stepan Chuprakov, Vladimir Gevorgyan

Research output: Contribution to journalArticlepeer-review

76 Scopus citations

Abstract

Figure presented It has been shown that various pyrido-, quinolino-, pyrazino-, and quinoxalinotetrazoles can be used efficiently as azide components in Cu-catalyzed click reaction with alkynes. This method allows for efficient synthesis of a wide variety of N-heterocyclic derivatives of 1,2,3-triazoles.

Original languageEnglish (US)
Pages (from-to)2166-2169
Number of pages4
JournalOrganic Letters
Volume12
Issue number9
DOIs
StatePublished - May 7 2010
Externally publishedYes

ASJC Scopus subject areas

  • Biochemistry
  • Physical and Theoretical Chemistry
  • Organic Chemistry

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