Synthesis and utility of dihydropyridine boronic esters

Santanu Panda, Aaron Coffin, Q. Nhu Nguyen, Dean J. Tantillo, Joseph M. Ready

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20 Scopus citations

Abstract

When activated by an acylating agent, pyridine boronic esters react with organometallic reagents to form a dihydropyridine boronic ester. This intermediate allows access to a number of valuable substituted pyridine, dihydropyridine, and piperidine products.

Original languageEnglish (US)
Pages (from-to)2205-2209
Number of pages5
JournalAngewandte Chemie - International Edition
Volume55
Issue number6
DOIs
Publication statusPublished - Feb 5 2016

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Keywords

  • allylic compounds
  • boron
  • heterocycles
  • samarium iodide
  • synthetic methods

ASJC Scopus subject areas

  • Chemistry(all)
  • Catalysis

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