Cu-catalyzed transannulation reaction of pyridotriazoles with terminal alkynes under aerobic conditions: Efficient synthesis of indolizines

V. Helan, A. V. Gulevich, V. Gevorgyan

Research output: Contribution to journalArticle

79 Citations (Scopus)

Abstract

A Cu(i)-catalyzed denitrogenative transannulation reaction of pyridotriazoles with terminal alkynes en route to indolizines was developed. Compared to the previously reported Rh-catalyzed transannulation reaction, this Cu-catalyzed method features aerobic conditions and a much broader scope of pyridotriazoles and alkynes.

Original languageEnglish (US)
Pages (from-to)1928-1931
Number of pages4
JournalChemical Science
Volume6
Issue number3
DOIs
StatePublished - Mar 1 2015
Externally publishedYes

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Indolizines
Alkynes

ASJC Scopus subject areas

  • Chemistry(all)

Cite this

Cu-catalyzed transannulation reaction of pyridotriazoles with terminal alkynes under aerobic conditions : Efficient synthesis of indolizines. / Helan, V.; Gulevich, A. V.; Gevorgyan, V.

In: Chemical Science, Vol. 6, No. 3, 01.03.2015, p. 1928-1931.

Research output: Contribution to journalArticle

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